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Ropsacitinib

    98%

Ropsacitinib

源葉(MedMol)
S20672
2127109-84-4
C20H17N9
383.41
Ropsacitinib;PF-06826647, Tyk2-IN-8
品牌 貨號(hào) 產(chǎn)品規(guī)格 價(jià)格(RMB) 庫(kù)存(上海) 北京 武漢 南京 購(gòu)買(mǎi)數(shù)量
源葉(MedMol) S20672-5mg 98% ¥1000.00元 4 - - -
源葉(MedMol) S20672-10mg 98% ¥1800.00元 5 - - -
源葉(MedMol) S20672-25mg 98% ¥3600.00元 5 - - -
源葉(MedMol) S20672-100mg 98% ¥9000.00元 預(yù)計(jì)交期:2-3天 - - -
產(chǎn)品介紹 參考文獻(xiàn) 質(zhì)檢證書(shū)(COA) 摩爾濃度計(jì)算器 相關(guān)產(chǎn)品

產(chǎn)品介紹

Ropsacitinib (PF-06826647, Tyk2-IN-8, compound 10) is a selective and orally administered inhibitor of tyrosine kinase 2 (TYK2) with IC50 of 17 nM for binding to TYK2 catalytically active JH1 domain. PF-06826647 (Tyk2-IN-8, compound 10) also inhibits JAK1 and JAK2 with IC50 of 383 nM and 74 nM, respectively. PF-06826647 (Tyk2-IN-8, compound 10) is used in the treatment of psoriasis (PSO).

產(chǎn)品描述:

Ropsacitinib (PF-06826647, Tyk2-IN-8, compound 10) is a selective and orally administered inhibitor of tyrosine kinase 2 (TYK2) with IC50 of 17 nM for binding to TYK2 catalytically active JH1 domain. PF-06826647 (Tyk2-IN-8, compound 10) also inhibits JAK1 and JAK2 with IC50 of 383 nM and 74 nM, respectively. PF-06826647 (Tyk2-IN-8, compound 10) is used in the treatment of psoriasis (PSO).

靶點(diǎn): TyrosineKinases
溶解性: soluble  in  DMSO
保存條件: -20℃
配置溶液濃度參考:
1mg 5mg 10mg
1 mM 2.608 ml 13.041 ml 26.082 ml
5 mM 0.522 ml 2.608 ml 5.216 ml
10 mM 0.261 ml 1.304 ml 2.608 ml
50 mM 0.052 ml 0.261 ml 0.522 ml
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參考文獻(xiàn)

質(zhì)檢證書(shū)(COA)

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批號(hào):JS298415 貨號(hào):S20001-25g
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摩爾濃度計(jì)算器

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