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PLURIPOTIN

    98%

Pluripotin

源葉(MedMol)
S81540
839707-37-8
C27H25F3N8O2
550.53
品牌 貨號 產(chǎn)品規(guī)格 價格(RMB) 庫存(上海) 北京 武漢 南京 購買數(shù)量
源葉(MedMol) S81540-2mg 98% ¥424.00元 5 - - -
源葉(MedMol) S81540-5mg 98% ¥640.00元 3 - - -
源葉(MedMol) S81540-10mg 98% ¥1160.00元 6 - - -
源葉(MedMol) S81540-25mg 98% ¥2240.00元 6 - - -
源葉(MedMol) S81540-50mg 98% ¥3520.00元 預(yù)計交期:2-3天 - - -
源葉(MedMol) S81540-100mg 98% ¥4960.00元 預(yù)計交期:2-3天 - - -
產(chǎn)品介紹 參考文獻 質(zhì)檢證書(COA) 摩爾濃度計算器 相關(guān)產(chǎn)品

產(chǎn)品介紹

Pluripotin is a dual inhibitor of ERK1 and RasGAP with KDs of 98 nM and 212 nM, respectively. Pluripotin also inhibits RSK1, RSK2, RSK3, and RSK4 with IC50s of 0.5, 2.5, 3.3, and 10.0 μM, respectively.
產(chǎn)品描述: Pluripotin is a dual inhibitor of ERK1 and RasGAP with KDs of 98 nM and 212 nM, respectively. Pluripotin also inhibits RSK1, RSK2, RSK3, and RSK4 with IC50s of 0.5, 2.5, 3.3, and 10.0 μM, respectively.
靶點: ERK1:98 nM (Kd);RasGAP:212 nM (Kd);RSK1:0.5 μM (IC50);RSK2:2.5 μM (IC50);RSK3:3.3 μM (IC50);RSK4:10 μM (IC50);ERK;?Raf;?S6Kinase
參考文獻: 1. Chen S, et al. Self-renewal of embryonic stem cells by a small molecule. Proc Natl Acad Sci U S A. 2006 Nov 14;103(46):17266-71. 2. Mertins SD, et al. A small molecule (pluripotin) as a tool for studying cancer stem cell biology: proof of concept. PLoS One. 2013;8(2):e57099.
溶解性: DMSO  :  25  mg/mL  (45.41  mM;  Need  ultrasonic)
保存條件: 2-8℃
配置溶液濃度參考:
1mg 5mg 10mg
1 mM 1.816 ml 9.082 ml 18.164 ml
5 mM 0.363 ml 1.816 ml 3.633 ml
10 mM 0.182 ml 0.908 ml 1.816 ml
50 mM 0.036 ml 0.182 ml 0.363 ml
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參考文獻

質(zhì)檢證書(COA)

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摩爾濃度計算器

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